2010 Apr;28(2):115-23. doi: 10.1007/s10637-009-9221-0. Epub 2009 Feb 3.
A metabolically stable analogue of anandamide, Met-F-AEA, inhibits human thyroid carcinoma cell lines by activation of apoptosis.
Abstract
![pm1](/wp-content/uploads/2013/04/Pub-Med-e1423848464246.jpg)
- PMID:
- 19189054
- [PubMed – indexed for MEDLINE]
-
Publication Types, MeSH Terms, Substances
Publication Types
MeSH Terms
- Apoptosis/drug effects*
- Arachidonic Acids/metabolism*
- Arachidonic Acids/pharmacology*
- Cell Cycle Proteins/metabolism
- Cell Line, Tumor
- Cell Nucleus/drug effects
- Cell Nucleus/metabolism
- Cell Proliferation/drug effects
- Drug Screening Assays, Antitumor
- Endocannabinoids
- Humans
- Molecular Weight
- Piperidines/pharmacology
- Poly(ADP-ribose) Polymerases/metabolism
- Polyunsaturated Alkamides/metabolism*
- Pyrazoles/pharmacology
- Receptor, Cannabinoid, CB1/antagonists & inhibitors
- Receptor, Cannabinoid, CB1/metabolism
- Thyroid Neoplasms/pathology*
- Tumor Suppressor Protein p53/metabolism
Substances
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