For Your Consideration... Ligand-Assisted Protein Structure (LAPS): An Experimental Paradigm for Characterizing Cannabinoid-Receptor Ligand-Binding Domains. Methods Enzymol. 2017;593:217-235. doi: 10.1016/bs.mie.2017.06.022. Epub 2017 Jul 3. Janero DR1, Korde A1, Makriyannis A2.…Freedom WaresJuly 3, 2017
Canna~Fangled Abstracts Leveraging allostery to improve G protein-coupled receptor (GPCR)-directed therapeutics: cannabinoid receptor 1 as a discovery target. 2016 Oct 7. Janero DR1, Thakur GA2. Author information Abstract INTRODUCTION: Allosteric modulators of G-protein coupled…Freedom WaresOctober 7, 2016